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Current Publications (2025)

1. A new phytopharmaceutical obtained from Polyalthia longifolia with anti-dyslipidemic potential: Mechanistic pathway insights exploiting co-inverse miRNA-mRNA expression analysis

Nilesh Khandelwal, Suriya Pratap Singh, Prashant Rai, Vinita Kushwaha, Sanchita Gupta, Astha Singh, Lorie Dehury, Amol Chhatrapati Bisen, Amrendra K Tiwari, Manish K Chourasia, Rabi Sankar Bhatta, Sudeep Tandon, Koneni V Sashidhara*, Anil N Gaikwad

Eur. J. Pharmacol., 991, 2025, 177297

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2. Design, synthesis and biological evaluation of new class of pyrazoles-dihydropyrimidinone derivatives as bone anabolic agents

Arvind Kumar Jaiswal, Anuj Raj, Ajay Kishor Kushawaha, Bhaskar Maji, Hemlata Bhatt, Shikha Verma, Sarita Katiyar, Alisha Ansari, Amol Chhatrapati Bisen, Arsh Tripathi, Mohammad Imran Siddiqi, Rabi Sankar Bhatta, Ritu Trivedi, Koneni V Sashidhara*

Bioorg. Chem., 157, 2025, 108216

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3. Design, synthesis, and biological evaluation of quinazolinone-dihydropyrimidinone as a potential anti-diabetic agent via GLUT4 translocation stimulation

Arvind Kumar Jaiswal, Ajay Kishor Kushawaha, Alisha Ansari, Nikita Chhikara, Sarita Katiyar, Ishbal Ahmad, Abhijit Deb Choudhury, Rabi Sankar Bhatta, Akhilesh K Tamrakar, Koneni V Sashidhara*

Eur. J. Med. Chem., 288, 2025, 117366

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4. Exploring Indole-Dihydropyrimidinone Derivatives: Design, Synthesis, Biological Assessment, SAR Analysis, and Evaluation of Mode of Action in Experimental Visceral Leishmaniasis

Garvita Mishra, Arvind Kumar Jaiswal, Ajay Kishor Kushawaha, Abhishek Kumar, Hemlata Bhatt, Alisha Ansari, Amol Chhatrapati Bisen, Rupa Hansda, Sristi Agrawal, Payel Acharjee, Rajdeep Guha, Rabi Sankar Bhatta, Bidyut Purkait, Koneni V. Sashidhara*

Eur. J. Med. Chem., 293, 2025, 117667

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5. Design, synthesis and evaluation of novel carboline-triazole hybrids as promising antimalarial agents

Rohini Nandi, Arvind Kumar Jaiswal, Hemlata Bhatt, Sarita Katiyar, Alisha Ansari, Abhijit Deb Choudhury, Shabeer Ali, Shikha Mishra, Rabi Sankar Bhatta, Mrigank Srivastava, Satish Mishra, Koneni V Sashidhara*

Eur. J. Med. Chem., 290, 2025, 117514

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6. Design, Synthesis, and Biological Evaluation of Isoxazole-Dihydropyrimidinone Hybrids as Potential Modulators of Adipogenesis and Dyslipidemia

Alisha Ansari, Nilesh Khandelwal, Jay Gupta, Prashant Rai, Arvind Kumar Jaiswal, Astha Singh, Sarita Katiyar, Ajay Kishor Kushawaha, Vinita Kushwaha, Anuradha Vishwakarma, Divyanshi Singh, Arpon Biswas, Ravi Kumar, Rabi Sankar Bhatta, Anil Nilkanth Gaikwad, Koneni V Sashidhara*

Eur. J. Med. Chem., 294, 2025, 117746

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7. Development of Novel Phthalazinone-Triazole Hybrids as Potential Antidiabetic Agents Targeting GLUT4 Translocation in Skeletal Muscle

Ajay Kishor Kushawaha, Arvind Kumar Jaiswal, Pawan Kumar, Sarita Katiyar, Rahul Baghel, Hemlata Bhatt, Jay Gupta, Alisha Ansari, Poonam Yadav, Ishbal Ahmad, Abhijit Deb Choudhury, Rabi Sankar Bhatta, Akhilesh K Tamrakar, Koneni V Sashidhara*

J. Med. Chem.2025

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Year wise publications

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