H index (50) Papers

Rare dipeptide and urea derivatives from roots of Moringa oleifera as potential anti-inflammatory and antinociceptive agents
Koneni V. Sashidhara*, Jammikuntla N. Rosaiah, Ethika Tyagi, Rakesh Shukla, Ram Raghubir, Siron M. Rajendran
European journal of medicinal chemistry, 2009, 44 (1), 432-436
Citations
184

Identification of quinoline-chalcone hybrids as potential antiulcer agents
Koneni V. Sashidhara*, Srinivasa Rao Avula, Vaibhav Mishra, Gopal Reddy Palnati, L. Ravithej Singh, Neetu Singh, Yashpal S. Chhonker, Priyanka Swami, R.S. Bhatta, Gautam Palit.
European journal of medicinal chemistry, 2015, 89, 638-653
Citations
129

Novel keto-enamine Schiffs bases from 7-hydroxy-4-methyl-2-oxo-2H-benzo [h] chromene-8, 10-dicarbaldehyde as potential antidyslipidemic and antioxidant agents
Koneni V. Sashidhara*, Jammikuntla N. Rosaiah, Gitika Bhatia, J.K. Saxena
European journal of medicinal chemistry, 2008, 43 (11), 2592-2596
Citations
101

16??Hydroxycleroda?3,13 (14)Z?dien?15,16?olide from�Polyalthia longifolia: a safe and orally active antileishmanial agent
Pragya Misra, Koneni V Sashidhara*, Suriya P. Singh, Awanish Kumar, Reema Gupta, Shailendra S Chaudhaery, Souvik Sen Gupta, HK Majumder, Anil K Saxena, Anuradha Dube*
British journal of pharmacology, 2010, 159 (5), 1143-1150
Citations
99

Novel Chalcone�Thiazole Hybrids as Potent Inhibitors of Drug Resistant�Staphylococcus aureus
Koneni V. Sashidhara*, K. Bhaskara Rao, Pragati Kushwaha, Ram K. Modukuri, Pratiksha Singh, Isha Soni, P. K. Shukla, Sidharth Chopra and Mukesh Pasupuleti.
ACS medicinal chemistry letters, 2013, 6 (7), 809-813
Citations
85

Discovery of coumarin�dihydropyridine hybrids as bone anabolic agents
Koneni V. Sashidhara*, Manoj Kumar, Vikram Khedgikar, Priyanka Kushwaha, Ram K. Modukuri, Abdhesh Kumar, Jyoti Gautam, Divya Singh, Balasubramaniam Sridhar, and Ritu Trivedi*
Journal of Medicinal Chemistry, 2013, 56 (1), 109-122
Citations
84

Synthesis and evaluation of novel triazolyl quinoline derivatives as potential antileishmanial agents
AkankshaUpadhyay, Pragati Kushwaha, SampaGupta, Ranga Prasad Dodda, Karthik Ramalingam, Ruchir Kant, NeenaGoyal, Koneni V.Sashidhara*
European Journal of Medicinal Chemistry, 2018, 154, 172-181
Citations
78

Antiplasmodial activity of novel keto-enamine chalcone-chloroquine based hybrid pharmacophores
Koneni V. Sashidhara*, Manoj Kumar, Ram K. Modukuri, Rajeev Kumar Srivastava, Awakash Soni, Kumkum Srivastava, Shiv Vardan Singh, J.K. Saxena, Harsh M. Gauniyal, Sunil K. Puri
Bioorganic & medicinal chemistry, 2012, 20 (9), 2971-2981
Citations
76

Design and synthesis of new series of coumarin�aminopyran derivatives possessing potential anti-depressant-like activity
Koneni V. Sashidhara *, Ram K. Modukuri, Seema Singh, K. Bhaskara Rao, G. Aruna Teja, Sampa Gupta, Shubha Shukla.
Bioorganic & Medicinal Chemistry Letters, 2015, 25 (2), 337-341
Citations
75

Coumarin�benzimidazole hybrids as a potent antimicrobial agent: synthesis and biological elevation
L. Ravithej Singh,Srinivasa Rao Avula, Sneha Raj, Akanksha Srivastava,Gopala Reddy Palnati, Tripathi CKM, Mukesh Pasupuleti*,Koneni V. Sashidhara*
The Journal of antibiotics, 2017, 70 (9), 954-961
Citations
73

The marine sponge metabolite mycothiazole: A novel prototype mitochondrial complex I inhibitor
J. Brian Morgan, Fakhri Mahdi, Yang Liu, Veena Coothankandaswamy, Mika B. Jekabsons, Tyler A. Johnson, Koneni V. Sashidhara, Phillip Crews, Dale G. Nagle*, Yu-Dong Zhou*
Bioorganic & medicinal chemistry, 2010, 18 (16), 5988-5994
Citations
70

Synthesis, Biological Evaluation, Structure?Activity Relationship and Mechanism of Action Studies of Quinoline-metronidazole Derivatives against Experimental Visceral Leishmaniasis
Akanksha Upadhyay, Pragya Chandrakar, Sampa Gupta, Naveen Parmar, Sandeep Kumar Singh, Mamunur Rashid, Pragati Kushwaha, M. Wahajuddin, Koneni V. Sashidhara* and Susanta Kar*
Journal of Medicinal Chemistry, 2019, 62 (11), 5655-5671
Citations
68

Isolation and identification of beta-hematin inhibitors from Flacourtia indica as promising antiplasmodial agents
Koneni V. Sashidhara*, Suriya P. Singh, Shiv Vardan Singh, Rajeev K. Srivastava, Kumkum Srivastava, J.K. Saxena, Sunil K. Puri
European journal of medicinal chemistry, 2013, 60, 497-502
Citations
67

Synthesis and bio-evaluation of indole-chalcone based benzopyrans as promising antiligase and antiproliferative agents
Sampa Gupta, Pooja Maurya, Akanksha Upadhyay, Pragati Kushwaha, Shagun Krishna, Mohammad Imran Siddiqi, Koneni V. Sashidhara*, Dibyendu Banerjee*
European journal of medicinal chemistry, 2018, 143, 1981-1996
Citations
62

Synthesis and in vitro evaluation of new chloroquine-chalcone hybrids against chloroquine-resistant strain of Plasmodium falciparum
Koneni V. Sashidhara*, Srinivasa Rao Avula, Gopala Reddy Palnati, Shiv Vardan Singh, Kumkum Srivastava, Sunil K. Puri, J.K. Saxena
Bioorganic & medicinal chemistry letters, 2012, 22 (17), 5455-5459
Citations
61

Neo-tanshinlactone inspired synthesis, in vitro evaluation of novel substituted benzocoumarin derivatives as potent anti-breast cancer agents
Koneni V. Sashidhara*, Jammikuntla N. Rosaiah, Manoj Kumar, Rishi Kumar Gara, Lakshma Vadithe Nayak, Kamini Srivastava, Hemant Kumar Bid, Rituraj Konwar
Bioorganic & medicinal chemistry letters, 2010, 20 (23), 7127-7131
Citations
61

Synthesis, biological evaluation and molecular dynamic simulations of novel Benzofuran-tetrazole derivatives as potential agents against Alzheimer�s disease
Pragati Kushwaha, Soobiya Fatima, Akanksha Upadhyay, Sampa Gupta, Sudha Bhagwati, TanviBaghel, M. I. Siddiqi, Aamir Nazir, Koneni V. Sashidhara*
Bioorganic & medicinal chemistry letters, 2019, 29 (1), 66-72
Citations
58

Cytotoxic cycloartane triterpene and rare isomeric bisclerodane diterpenes from the leaves of Polyalthia longifolia var. pendula
Koneni V. Sashidhara*, Suriya P. Singh, Ruchir Kant, Prakas R. Maulik, Jayanta Sarkar, Sanjeev Kanojiya, K. Ravi Kumar
Bioorganic & medicinal chemistry letters, 2010, 20 (19), 5767-5771
Citations
57

Discovery of a new class of HMG-CoA reductase inhibitor from Polyalthia longifolia as potential lipid lowering agent
Koneni V. Sashidhara*, Suriya P. Singh, Anuj Srivastava, Anju Puri, Yashpal S. Chhonker, Rabi S. Bhatta, Priyanka Shah, Mohammad Imran Siddiqi










