2018 Publications

1. In-house chemical library repurposing: A case example for Pseudomonas aeruginosa antibiofilm activity and quorum sensing inhibition

L Ravithej Singh, Vikash C Tripathi, Sneha Raj, Anoop Kumar, Sampa Gupta, Soyar Horam, Akanksha Upadhyay, Pragati Kushwaha, Jesu Arockiaraj, Koneni V Sashidhara, Mukesh Pasupuleti

Drug Dev. Res., 79, 2018, 383-390

2. Pharmacokinetics, metabolism, bioavailability, tissue distribution and excretion studies of 16α-hydroxycleroda-3, 13(14) Z -dien-15, 16-olide—a novel HMG-CoA reductase inhibitor

Tulsankar Sachin Laxman, Santosh Kumar Puttrevu, Rajesh Pradhan, Anjali Mishra, Sarvesh Verma, Yashpal S Chhonker, Swarnim Srivastava, Suriya P Singh, Koneni V Sashidhara, Rabi Sankar Bhatta

Naunyn-Schmiedeberg's Arch. Pharmacol., 391, 2018, 965-973

3. Synthesis and study of benzofuran-pyran analogs as BMP-2 targeted osteogenic agents

Pragati Kushwaha, Ashish Kumar Tripathi, Sampa Gupta, Priyanka Kothari, Akanksha Upadhyay, Naseer Ahmad, Tanuj Sharma, MI Siddiqi, Ritu Trivedi, Koneni V Sashidhara*

Eur. J. Med. Chem., 156, 2018, 103-117

4. Synthesis and evaluation of novel triazolyl quinoline derivatives as potential antileishmanial agents

Akanksha Upadhyay, Pragati Kushwaha, Sampa Gupta, Ranga Prasad Dodda, Karthik Ramalingam, Ruchir Kant, Neena Goyal, Koneni V Sashidhara*

Eur. J. Med. Chem., 154, 2018, 172-181

5. Benzofuran-pyran hybrids: A new class of potential bone anabolic agents

Sampa Gupta, Sulekha Adhikary, Ram K Modukuri, Dharmendra Choudhary, Ritu Trivedi, Koneni V Sashidhara*

Bioorg. Med. Chem. Lett., 28, 2018, 1719-1724

6. Discovery of coumarin-dihydroquinazolinone analogs as niacin receptor 1 agonist with in-vivo anti-obesity efficacy

L Ravithej Singh, Ajeet Kumar, Akanksha Upadhyay, Sampa Gupta, Gopala Reddy Palanati, Kamakshi Sikka, Mohammad Imran Siddiqi, Prem N Yadav, Koneni V Sashidhara*

Eur. J. Med. Chem., 152, 2018, 208-222

7. Overexpression of DNA ligase I compensates for Topoisomerase I inhibition leading to resistance in human colorectal cancer cells

P Maurya, S Gupta, S Krishna, MI Siddiqi, KV Sashidhara, D Banerjee

Cancer Medicine, 7, 2018, 15

8. Substituted carbamothioic amine-1-carbothioic thioanhydrides as novel trichomonicidal fungicides: Design, synthesis, and biology

Dhanaraju Mandalapu, Bhavana Kushwaha, Sonal Gupta, Shagun Krishna, Nidhi Srivastava, Mahendra Shukla, Pratiksha Singh, Bhavana S Chauhan, Ravi Goyani, Jagdamba P Maikhuri, Koneni V Sashidhara, Brijesh Kumar, Renu Tripathi, Praveen K Shukla, Mohammad I Siddiqi, Jawahar Lal, Gopal Gupta, Vishnu L Sharma

Eur. J. Med. Chem., 143, 2018, 632-645

9. Synthesis and bio-evaluation of indole-chalcone based benzopyrans as promising antiligase and antiproliferative agents

Sampa Gupta, Pooja Maurya, Akanksha Upadhyay, Pragati Kushwaha, Shagun Krishna, Mohammad Imran Siddiqi, Koneni V Sashidhara, Dibyendu Banerjee

Eur. J. Med. Chem., 143, 2018, 1981-1996

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